Abstract
A novel benzimidazole series of small-molecule thrombopoietin receptor agonists has been discovered. Herein, we discuss the preliminary exploration of structure-activity relationships within this chemotype.
MeSH terms
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Acids / chemistry
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Benzimidazoles / chemical synthesis
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Benzimidazoles / chemistry*
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Benzimidazoles / pharmacology*
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Molecular Structure
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Naphthols / chemistry
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Receptors, Cytokine / agonists*
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Receptors, Cytokine / metabolism*
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Structure-Activity Relationship
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Thrombopoietin / metabolism*
Substances
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Acids
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Benzimidazoles
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Naphthols
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Receptors, Cytokine
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Thrombopoietin
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benzimidazole